{"id":1225,"date":"2022-10-03T12:54:40","date_gmt":"2022-10-03T12:54:40","guid":{"rendered":"https:\/\/flmodafinil.pl\/sklep\/coluracetam-purete-de-la-substance-%e2%89%a5-99-1000mg\/"},"modified":"2022-10-29T20:30:26","modified_gmt":"2022-10-29T20:30:26","slug":"coluracetam","status":"publish","type":"product","link":"https:\/\/flmodafinil.pl\/fr\/sklep\/coluracetam\/","title":{"rendered":"Coluracetam, puret\u00e9 de la substance \u2265 99%, 1000mg"},"content":{"rendered":"<h1>Coluracetam 1000 mg<\/h1>\n<ul>\n<li>\n<h5>Puret\u00e9 \u2265 99%<\/h5>\n<\/li>\n<li>\n<h5>Poids net : 1 gramme<\/h5>\n<\/li>\n<li>\n<h5>Num\u00e9ro CAS : 135463-81-9<\/h5>\n<\/li>\n<li>\n<h5>Formule mol\u00e9culaire : C19H23N3O3<\/h5>\n<\/li>\n<li>\n<h5>Poids mol\u00e9culaire : 341,411 g-mol-1<\/h5>\n<\/li>\n<li>\n<h5>Forme : Poudre<\/h5>\n<\/li>\n<\/ul>\n<h5>Description de la Wikip\u00e9dia anglaise :<\/h5>\n<h6>Le coluracetam (DCI ; code de d\u00e9veloppement BCI-540 ; anciennement MKC-231) est un agent nootrope putatif de la famille des rac\u00e9tams[1]. Il contient un groupe chimique qui est un bioisost\u00e8re de la famille des 9-amino-t\u00e9trahydroacridines. Il a \u00e9t\u00e9 initialement d\u00e9velopp\u00e9 et test\u00e9 par Mitsubishi Tanabe Pharma Corporation pour la maladie d&rsquo;Alzheimer. Apr\u00e8s que le m\u00e9dicament n&rsquo;ait pas atteint les objectifs fix\u00e9s lors des essais cliniques, BrainCells Inc. en a obtenu la licence pour mener des recherches sur le trouble d\u00e9pressif majeur (TDM), qui ont \u00e9t\u00e9 pr\u00e9c\u00e9d\u00e9es d&rsquo;une \u00ab\u00a0subvention de programme de d\u00e9couverte th\u00e9rapeutique qualifiante\u00a0\u00bb de l&rsquo;\u00c9tat de Californie. 2] Les r\u00e9sultats d&rsquo;essais cliniques de phase IIa sugg\u00e8rent qu&rsquo;il s&rsquo;agirait d&rsquo;un traitement potentiel pour le TDM comorbide avec trouble anxieux g\u00e9n\u00e9ralis\u00e9 (TAG)[3]. BrainCells Inc. est en train de retirer le m\u00e9dicament \u00e0 cette fin ( [kiedy?] ). [4] [wymagane pe\u0142ne cytowanie] Il pourrait \u00e9galement avoir une utilisation potentielle dans la pr\u00e9vention et le traitement de la r\u00e9tinopathie isch\u00e9mique et des l\u00e9sions de la r\u00e9tine et du nerf optique.  [wymagane cytowanie medyczne]<\/h6>\n<h6>Il a \u00e9t\u00e9 d\u00e9montr\u00e9 que le <a href=\"https:\/\/flmodafinil.pl\/coluracetam-poprawia-prace-mozgu-lagodzi-stany-depresyjne\/\">coluracetam<\/a> inverse la perte de production de choline ac\u00e9tyltransf\u00e9rase dans le noyau septal m\u00e9dian de rats expos\u00e9s \u00e0 la phencyclidine (PCP) et est consid\u00e9r\u00e9 comme un m\u00e9dicament th\u00e9rapeutique potentiel pour la schizophr\u00e9nie.<\/h6>\n<h6>Le coluracetam augmente le captage de choline de haute affinit\u00e9 (HACU) [6], qui est l&rsquo;\u00e9tape limitant la vitesse de synth\u00e8se de l&rsquo;ac\u00e9tylcholine (ACh). Des \u00e9tudes ont montr\u00e9 que le coluracetam am\u00e9liore les troubles de l&rsquo;apprentissage apr\u00e8s une dose orale unique administr\u00e9e \u00e0 des rats expos\u00e9s \u00e0 des neurotoxines cholinergiques. Des \u00e9tudes ult\u00e9rieures ont montr\u00e9 qu&rsquo;il peut induire des effets pro-cognitifs \u00e0 long terme chez des rats trait\u00e9s par des neurotoxines cholinergiques en modifiant le syst\u00e8me de r\u00e9gulation du transporteur de choline.[7]Produit r\u00e9serv\u00e9 \u00e0 un usage en laboratoire. Non destin\u00e9 \u00e0 la consommation.<\/h6>\n<p>Pour en savoir plus sur le Coulracetam, lisez l&rsquo;article en polonais :<\/p>\n<blockquote class=\"wp-embedded-content\" data-secret=\"HlmJahNCtm\"><p><a href=\"https:\/\/flmodafinil.pl\/coluracetam-poprawia-prace-mozgu-lagodzi-stany-depresyjne\/\">Coluracetam &#8211; poprawia prac\u0119 m\u00f3zgu, \u0142agodzi stany depresyjne<\/a><\/p><\/blockquote>\n<p><iframe loading=\"lazy\" class=\"wp-embedded-content\" sandbox=\"allow-scripts\" security=\"restricted\" style=\"position: absolute; clip: rect(1px, 1px, 1px, 1px);\" title=\"\u00ab\u00a0Coluracetam &#8211; poprawia prac\u0119 m\u00f3zgu, \u0142agodzi stany depresyjne\u00a0\u00bb &#8212; NONSENSIA, Laboratorium.\" src=\"https:\/\/flmodafinil.pl\/coluracetam-poprawia-prace-mozgu-lagodzi-stany-depresyjne\/embed\/#?secret=4aEZObPDH7#?secret=HlmJahNCtm\" data-secret=\"HlmJahNCtm\" width=\"600\" height=\"338\" frameborder=\"0\" marginwidth=\"0\" marginheight=\"0\" scrolling=\"no\"><\/iframe><\/p>\n<p>&nbsp;<\/p>\n","protected":false},"excerpt":{"rendered":"<p>Coluracetam produit chimique pur de la famille des racetams disponible \u00e0 l&rsquo;achat en ligne. Le profil du coluracetam est une affinit\u00e9 \u00e9lev\u00e9e pour la choline.<\/p>\n","protected":false},"featured_media":607,"template":"","meta":[],"product_brand":[],"product_cat":[197],"product_tag":[670,664,669,661,667,672,671],"class_list":["post-1225","product","type-product","status-publish","has-post-thumbnail","product_cat-non-classe","product_tag-absorption-de-la-choline","product_tag-bci-540-fr","product_tag-c19h23n3o3-fr","product_tag-coluracetam-fr","product_tag-mkc-231-fr","product_tag-numero-de-cas-135463-81-9-fr","product_tag-tricyanoaminopropene-fr","first","instock","shipping-taxable","purchasable","product-type-variable"],"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.9 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Coluracetam, puret\u00e9 de la substance \u2265 99%, 1000mg - NONSENSIA, Laboratorium.<\/title>\n<meta name=\"description\" content=\"Coluracetam produit chimique pur de la famille des racetams disponible \u00e0 l&#039;achat en ligne. 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